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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T14391 Azidamfenicol

Antibacterial; Antibiotic Microbiology/Virology
Azidamfenicol 抑制核糖体肽基转移酶,Ki 为 22 µM。Azidamfenicol 是一种广谱氯霉素类抗生素。
T4998L Cefpodoxime (free acid)

Others Others
Cefpodoxime (free acid) 是一种口服的第三代头孢菌素抗生素。除铜绿假单胞菌、肠球菌和脆弱拟杆菌外,它对大多数革兰氏阳性和革兰氏阴性微生物均有效。
T9680 Irloxacin

Antibacterial Microbiology/Virology
Irloxacin 是一种口服活性的喹诺酮类抗菌剂,在酸性条件下具有更强大的活性。在体外,Irloxacin 对革兰氏阳性菌和革兰氏阴性菌都具有良好的抗菌谱。
T20525 Chloramphenicol palmitate

Antibacterial; Antibiotic Microbiology/Virology
Chloramphenicol palmitate 是一种广谱抗生素,对革兰氏阳性和革兰氏阴性细菌具有活性。 Chloramphenicol palmitate 可用于在含有氯霉素抗性基因的转化细胞中作为细菌选择剂的研究。
T1008 Cephalexin

头孢氨苄,Cefalexin,Cephacillin

Antibacterial; Antibiotic Microbiology/Virology
Cephalexin (Cephacillin) 是一种强口服活性的头孢菌素抗生素。它通过破坏细菌细胞壁的生长来杀死革兰氏阳性和一些革兰氏阴性细菌。它可研究肺炎、链球菌性咽喉炎、细菌性心内膜炎等。
T5006 Flucloxacillin sodium

氟氯西林钠,floxacillin sodium

Antibacterial; Antibiotic Microbiology/Virology
Flucloxacillin sodium (floxacillin sodium) 是一种高活性抗生素,抑制革兰氏阳性和革兰氏阴性菌。
T6582 Mezlocillin Sodium

美洛西林钠,Baycipen

Antibacterial; Antibiotic Microbiology/Virology
Mezlocillin Sodium (Baycipen) 是一种青霉素 β-内酰胺类抗生素,用于治疗由易感染微生物引起的细菌感染。
T3117 Marbofloxacin

马波沙星,Marbofloxacine,Zeniquin,Marbocyl

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Marbofloxacin (Zeniquin) 是一种具有口服活性的氟喹诺酮类广谱抗菌剂。它可研究革兰氏阳性和革兰氏阴性细菌以及支原体引起的感染。
TP1444 Magainin 2

蛙皮素 2

Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Magainin 2是从非洲爪蟾皮肤中分离得到的一种抗菌肽。它对许多革兰氏阴性和革兰氏阳性细菌显示出抗生素活性,对原生动物也有活性。它通过优先与细菌膜中丰富的阴离子磷脂相互作用而发挥细胞毒性作用。
T0396 Pipemidic acid

吡哌酸,Acido pipemidico

Antibacterial; Antibiotic Microbiology/Virology
Pipemidic acid (Acido pipemidico) 是一种新型抗菌剂,对革兰氏阴性菌和某些革兰氏阳性细菌具有活性,可研究肠道、泌尿和胆道感染。
T0116 Balofloxacin

DNA gyrase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Balofloxacin 是一种具有口服活性的氟喹诺酮类抗生素,可通过干扰 DNA 促旋酶来抑制细菌 DNA 的合成,对革兰氏阴性,革兰氏阳性和厌氧菌具有广谱抗菌活性。它可研究呼吸道,肠道和泌尿道感染。
T9066 Merafloxacin

CI 934

SARS-CoV Microbiology/Virology
Merafloxacin (CI 934) 是一种氟喹诺酮类抗菌药物,也被确定为 SARS-CoV-2 的 1 PRF 抑制剂。它对革兰氏阳性菌和革兰氏阴性菌具有体外活性。
T7865 Danofloxacin

达氟沙星,达诺沙星,Danofloxacino,Danofloxacin free base,Danofloxacine

Others; DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others
Danofloxacin (Danofloxacin free base) free base 是一种具有口服活性第三代氟喹诺酮抗菌剂,对大多数革兰氏阴性和革兰氏阳性细菌,支原体和衣原体物种具有广谱的活性,并通过抑制细菌的 DNA 回转酶发挥抗菌作用。它可用于牛,猪和鸡呼吸道疾病的研究。
T2692 A40926

Dalbavancin Impurity,达巴霉素杂质

Antibacterial Microbiology/Virology
A40926 (Dalbavancin Impurity) 是Dalbavancin 的前体,是一种糖肽抗生素。它抑制革兰氏阳性细菌,对淋病奈瑟氏球菌非常有效。
T0133 Cefdinir

FK-482,头孢地尼,CI-983,PD 134393

Glutathione Peroxidase; Antibacterial; Antibiotic Metabolism; Microbiology/Virology
Cefdinir (FK-482) 是头孢菌素类中的一种半合成广谱抗生素,对几种革兰氏阴性和革兰氏阳性细菌引起的感染有效。它可研究耳,鼻窦,喉咙和皮肤的常见细菌感染。
T73997 Anti gram-positive/negative bacteria agent 1

Anti gram-positive/negative bacteria agent 1 是一种含有基于MECAM的人工铁载体的抗生素化合物。
T20774 Sarafloxacin

A-56620,A 56620,A56620,沙拉沙星

Antibacterial; Antibiotic Microbiology/Virology
Sarafloxacin (A56620) 对革兰氏阳性菌和革兰氏阴性菌具有抗菌活性。
T1640 Ciprofloxacin

Ciproxan,环丙沙星,Ciprobay,Bay o 9867,Bay-09867

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Ciprofloxacin (Bay-09867) 是一种有高抗菌活性的氟喹诺酮类抗生素。
T11315 Fosmidomycin sodium salt

FR-31564 sodium salt

Antibiotic; Parasite Microbiology/Virology
Fosmidomycin sodium salt (FR-31564 sodium salt) 是一种抗感染类抗生素,具有抗疟疾活性,抑制革兰氏阴性菌和革兰氏阳性菌。
T11301L Flomoxef sodium

Others Others
Flomoxef sodium 属于奥沙环类抗生素,对多种革兰氏阳性菌均具有良好的杀灭活性。
T0425 Pefloxacin Mesylate

Pefloxacinium mesylate,甲磺酸培氟沙星

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Pefloxacin Mesylate (Pefloxacinium mesylate) 是一种抗菌化合物,可抑制DNA 旋转酶阻断DNA 复制。
T11123 DuP 105

Antibacterial; Antibiotic Microbiology/Virology
DuP 105是可口服的oxazolidinone类化合物,这是一种新型合成的抗菌化合物,对革兰氏阳性细菌具有有效性。
T6706 Ticarcillin sodium

Ticarpen hydrate,Aerugipen hydrate,替卡西林单钠盐单水合物,BRL 2288,AB 2288,Monapen

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Ticarcillin sodium (Aerugipen hydrate) 主要用于抗革兰氏阴性菌, 也能用于研究嗜麦芽感染。
TP1763L Magainin 1 acetate

Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Magainin 1 acetate 是一种抗菌肽。它对许多革兰氏阴性和革兰氏阳性细菌表现出抗生素活性。
T4020 Cadazolid

ACT-179811,卡达唑利德

Antibacterial; Antibiotic Microbiology/Virology
Cadazolid (ACT-179811) 是一种新型恶唑烷酮类抗生素,对Clostridium difficile 有活性。
T73054 Moiramide B

Acetyl-CoA Carboxylase; Antibiotic Metabolism; Microbiology/Virology
Moiramide B 是一种高效的乙酰辅酶 A 羧化酶 (ACC) 抑制剂(IC50:6 nM),具有抗菌活性,强烈抑制革兰氏阳性菌,但对革兰氏阴性菌的抑制效果较弱。
TP1663L CysHHC10 acetate

CysHHC10 acetate(1408311-03-4 free base)

Antibacterial Microbiology/Virology
CysHHC10 acetate 对革兰氏阳性菌和革兰氏阴性菌均具有抗菌活性,对大肠杆菌、铜绿假单胞菌、金黄色葡萄球菌和表皮葡萄球菌的 MIC 分别为 10.1、20.2、2.5 和 1.3 mM。
T28229 Olanexidine hydrochloride

OPB2045,OPB-2045,OPB-2045 HCl,OPB 2045

Antibacterial Microbiology/Virology
Olanexidine hydrochloride (OPB-2045 HCl) 对革兰氏阳性菌和革兰氏阴性菌具有杀菌活性。 Olanexidine hydrochloride 破坏金黄色葡萄球菌的膜完整性。
T0967 Teicoplanin

Antibiotic MDL-507,MDL-507,替考拉宁,Teichomycin

Antibacterial; Antibiotic Microbiology/Virology
Teicoplanin (MDL-507) 是一种半合成的糖肽抗生素, 可用于由革兰氏阳性菌引起的严重感染的相关研究。
T22228 Tylvalosin tartrate

酒石酸乙酰异戊酰泰乐菌素,Acetylisovaleryltylosin Tartrate

Antibacterial; Antibiotic Microbiology/Virology
Tylvalosin tartrate (Acetylisovaleryltylosin Tartrate) 是一种对革兰氏阳性细菌具有抗性的大环内酯类抗生素。
T17021 Tebipenem

LJC 11036

Antibiotic Microbiology/Virology
Tebipenem 是一种口服碳青霉烯类抗生素。 它对革兰氏阳性和阴性细菌具有广谱活性。
T3247 Lysozyme from chicken egg white

鸡蛋清溶菌酶,溶菌酶,Lysozyme

Others; Antibacterial Microbiology/Virology; Others
Lysozyme from chicken egg white (Lysozyme) 是一种存在于鸡蛋清中的杀菌酶,它溶解革兰氏阳性菌。
T0897 Nitrofurazone

NFZ,呋喃西林,Nitrofural,Furacilin

Dehydrogenase; Antibacterial; Glutathione reductase; Antibiotic Metabolism; Microbiology/Virology; oxidation-reduction
Nitrofurazone (Furacilin) 是一种抗生素。
T19709 Nitrocefin

Others Others
Nitrocefin 是 β-内酰胺酶的显色底物,当 β-内酰胺酶将 β-内酰胺环中的酰胺键水解后,Nitrocefin 的颜色会由黄色变为红色。它可用于 β-内酰胺酶耐药抗生素的研究。
T19860 Clavulanic Acid

BRL 14151,MM-14151,MM 14151,RX-10100,MM14151,BRL14151,BRL-14151

Antibacterial; Antifungal Microbiology/Virology
Clavulanic Acid(RX-10100) 是一种由生物体克拉维链霉菌产生的主要β-内酰胺类抗生素,是一种强效的细菌 β-内酰胺酶抑制剂,用于研究细菌引起的感染。Clavulanic Acid 具有广谱的生物活性,对多种革兰氏阳性和革兰氏阴性细菌均有活性。
T1001 Dicloxacillin Sodium hydrate

Dicloxacillin sodium salt monohydrate,双氯西林钠,Dicloxacillin sodium monohydrate

Antibacterial; Antibiotic Microbiology/Virology
Dicloxacillin Sodium hydrate 是一种青霉素类窄谱β内酰胺抗生素,可研究革兰氏阳性菌感染。
T22408 Proflavine

吡啶-3,6-二胺,3,6-Diaminoacridine

Antibacterial Microbiology/Virology
Proflavine (3,6-Diaminoacridine) 是吖啶染料,可用作抗菌剂。它是 DNA 嵌入剂,能够阻滞Kir3.2孔。它用作与 Kir3.2 相关的神经系统疾病的研究。
T68137 Sanfetrinem

GV104326

Antibiotic Microbiology/Virology
Sanfetrinem (GV104326) sodium 是一种新型可口服 β-内酰胺酶抗生素,对革兰氏阳性菌和革兰氏阴性菌显示出显著的抗菌活性,可用于研究细菌感染。
T7043 Cefotetan

头孢替坦,Apacef

Antibacterial; Antibiotic Microbiology/Virology
Cefotetan (Apacef) 是一种半合成的头霉素抗生素,能抑制细胞壁合成发挥杀菌作用。
T1492 Gemifloxacin mesylate

LB-20304a,甲磺酸吉米沙星,SB-265805S,Gemifloxacin mesylate

DNA gyrase; Topoisomerase; Antibacterial DNA Damage/DNA Repair; Microbiology/Virology
Gemifloxacin mesylate (Gemifloxacin mesylate) 是一种喹诺酮类口服广谱抗菌剂,可研究轻中度肺炎和慢性支气管炎的急性细菌性发作。
T14951 Chlorhexidine digluconate

Apoptosis; Antibiotic Apoptosis; Microbiology/Virology
Chlorhexidine digluconate 是一种广谱防腐剂和消毒剂,具有广谱抗菌活性,抑制革兰氏阳性菌和革兰氏阴性菌,可诱导细胞坏死和凋亡,可用于研究细菌感染。
T22391 Omeprazole Sodium

P450; Proton pump; Antibacterial; Autophagy Autophagy; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology
Omeprazole 是有效的质子泵抑制剂,在胃肠道疾病的研究中具有价值。它竞争性抑制CYP2C19活性,Ki 为 2 到 6 μM。它还抑制革兰氏阴性菌和革兰氏阳性菌生长。它是中性鞘磷脂酶的外泌体抑制剂。
T4998 Cefpodoxime proxetil

Antibacterial; Antibiotic Microbiology/Virology
Cefpodoxime Proxetil 是一种口服的广谱型抗生素。它与青霉素结合蛋白结合,抑制肽聚糖的合成,干扰细菌细胞壁的生物合成。
T9449 Nitrofural

[(E)-(5-nitrofuran-2-yl)methylideneamino,(E)-2-((5-硝基呋喃-2-基)亚甲基)肼甲酰胺

Antibacterial Microbiology/Virology
Nitrofural 是 20 世纪已在临床应用中确立的硝基呋喃。 Nitrofural 在临床上对广泛的革兰氏阳性和革兰氏阴性细菌(包括许多常见的泌尿道病原体菌株)仍然有效。
T0195 Secnidazole

RP-14539,PM-185184,塞克硝唑

Antibiotic; Parasite Microbiology/Virology
Secnidazole (PM-185184) 是一种具有口服活性唑类抗生素,半衰期比甲硝唑更长。它有潜力研究细菌性阴道病。
T7858 Ceftezole sodium

Celoslin,Falomesin,头孢替唑钠,Alomen

Anti-infection; Antibacterial; Antibiotic; Glucosidase Metabolism; Microbiology/Virology
Ceftezole sodium (Falomesin) 是一种广谱 cephem 抗生素,具有抑制多种革兰氏阳性菌和革兰氏阴性菌活性。它是一种α-葡萄糖苷酶抑制剂,具有体内抗糖尿病活性。
T0932 Cefixime

FK-027,头孢克肟,Cefspan,Cefiximum,Cephoral,FR-17027,CL-284635

Antibacterial; Antibiotic Microbiology/Virology
Cefixime (FR-17027) 是一种头孢菌素类抗生素, 可研究一些细菌感染。
T1060 Flumequine

Flumigal,氟甲喹,R-802

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Flumequine (R-802) 是一种喹诺酮类抗生素,对革兰氏阳性菌和革兰氏阴性菌均有效。它是拓扑异构酶 II 抑制剂, 抑制细胞分裂,IC50值为 15 μM (3.92 μg/mL)。
T0911 Cefotaxime sodium

Cefotaxim sodium salt,头孢噻肟钠,Cefotaxime sodium salt,Cefotaxim (sodium salt),HR-756 (sodium salt)

Antibacterial; Antibiotic Microbiology/Virology
Cefotaxime sodium (Cefotaxim sodium salt) 是头孢类抗生素和耐内酰胺酶的头孢菌素,有抗革兰氏阳性菌和革兰氏阴性菌作用。
T124492 Imipenem

N-Formimidoyl thienamycin,MK0787

Antifungal Microbiology/Virology
Imipenem (MK0787) 是一种噻吩霉素衍生物,属于抗生素类,具有抗菌活性,对革兰氏阳性和革兰氏阴性菌具有部分的抑制作用。Imipenem 可用于研究碳青霉烯类非易感性感染和铜绿假单胞菌生物膜感染。

化合物

Azidamfenicol
Cat.No: T14391
Synonym:
Target: Antibacterial, Antibiotic
Cefpodoxime (free acid)
Cat.No: T4998L
Synonym:
Target: Others
Irloxacin
Cat.No: T9680
Synonym:
Target: Antibacterial
Chloramphenicol palmitate
Cat.No: T20525
Synonym:
Target: Antibacterial, Antibiotic
Cephalexin
Cat.No: T1008
Synonym: 头孢氨苄,Cefalexin,Cephacillin
Target: Antibacterial, Antibiotic
Flucloxacillin sodium
Cat.No: T5006
Synonym: 氟氯西林钠,floxacillin sodium
Target: Antibacterial, Antibiotic
Mezlocillin Sodium
Cat.No: T6582
Synonym: 美洛西林钠,Baycipen
Target: Antibacterial, Antibiotic
Marbofloxacin
Cat.No: T3117
Synonym: 马波沙星,Marbofloxacine,Zeniquin,Marbocyl
Target: Topoisomerase, Antibacterial, Antibiotic
Magainin 2
Cat.No: TP1444
Synonym: 蛙皮素 2
Target: Antibacterial, Antibiotic, Antifungal
Pipemidic acid
Cat.No: T0396
Synonym: 吡哌酸,Acido pipemidico
Target: Antibacterial, Antibiotic
Balofloxacin
Cat.No: T0116
Synonym:
Target: DNA gyrase, Antibacterial, Antibiotic
Merafloxacin
Cat.No: T9066
Synonym: CI 934
Target: SARS-CoV
Danofloxacin
Cat.No: T7865
Synonym: 达氟沙星,达诺沙星,Danofloxacino,Danofloxacin free base,Danofloxacine
Target: Others, DNA/RNA Synthesis, Antibacterial, Antibiotic
A40926
Cat.No: T2692
Synonym: Dalbavancin Impurity,达巴霉素杂质
Target: Antibacterial
Cefdinir
Cat.No: T0133
Synonym: FK-482,头孢地尼,CI-983,PD 134393
Target: Glutathione Peroxidase, Antibacterial, Antibiotic
Anti gram-positive/negative bacteria agent 1
Cat.No: T73997
Synonym:
Target:
Sarafloxacin
Cat.No: T20774
Synonym: A-56620,A 56620,A56620,沙拉沙星
Target: Antibacterial, Antibiotic
Ciprofloxacin
Cat.No: T1640
Synonym: Ciproxan,环丙沙星,Ciprobay,Bay o 9867,Bay-09867
Target: Topoisomerase, Antibacterial, Antibiotic
Fosmidomycin sodium salt
Cat.No: T11315
Synonym: FR-31564 sodium salt
Target: Antibiotic, Parasite
Flomoxef sodium
Cat.No: T11301L
Synonym:
Target: Others
Pefloxacin Mesylate
Cat.No: T0425
Synonym: Pefloxacinium mesylate,甲磺酸培氟沙星
Target: Topoisomerase, Antibacterial, Antibiotic
DuP 105
Cat.No: T11123
Synonym:
Target: Antibacterial, Antibiotic
Ticarcillin sodium
Cat.No: T6706
Synonym: Ticarpen hydrate,Aerugipen hydrate,替卡西林单钠盐单水合物,BRL 2288,AB 2288,Monapen
Target: Others, Antibacterial, Antibiotic
Magainin 1 acetate
Cat.No: TP1763L
Synonym:
Target: Antibacterial, Antibiotic, Antifungal
Cadazolid
Cat.No: T4020
Synonym: ACT-179811,卡达唑利德
Target: Antibacterial, Antibiotic
Moiramide B
Cat.No: T73054
Synonym:
Target: Acetyl-CoA Carboxylase, Antibiotic
CysHHC10 acetate
Cat.No: TP1663L
Synonym: CysHHC10 acetate(1408311-03-4 free base)
Target: Antibacterial
Olanexidine hydrochloride
Cat.No: T28229
Synonym: OPB2045,OPB-2045,OPB-2045 HCl,OPB 2045
Target: Antibacterial
Teicoplanin
Cat.No: T0967
Synonym: Antibiotic MDL-507,MDL-507,替考拉宁,Teichomycin
Target: Antibacterial, Antibiotic
Tylvalosin tartrate
Cat.No: T22228
Synonym: 酒石酸乙酰异戊酰泰乐菌素,Acetylisovaleryltylosin Tartrate
Target: Antibacterial, Antibiotic
Tebipenem
Cat.No: T17021
Synonym: LJC 11036
Target: Antibiotic
Lysozyme from chicken egg white
Cat.No: T3247
Synonym: 鸡蛋清溶菌酶,溶菌酶,Lysozyme
Target: Others, Antibacterial
Nitrofurazone
Cat.No: T0897
Synonym: NFZ,呋喃西林,Nitrofural,Furacilin
Target: Dehydrogenase, Antibacterial, Glutathione reductase, Antibiotic
Nitrocefin
Cat.No: T19709
Synonym:
Target: Others
Clavulanic Acid
Cat.No: T19860
Synonym: BRL 14151,MM-14151,MM 14151,RX-10100,MM14151,BRL14151,BRL-14151
Target: Antibacterial, Antifungal
Dicloxacillin Sodium hydrate
Cat.No: T1001
Synonym: Dicloxacillin sodium salt monohydrate,双氯西林钠,Dicloxacillin sodium monohydrate
Target: Antibacterial, Antibiotic
Proflavine
Cat.No: T22408
Synonym: 吡啶-3,6-二胺,3,6-Diaminoacridine
Target: Antibacterial
Sanfetrinem
Cat.No: T68137
Synonym: GV104326
Target: Antibiotic
Cefotetan
Cat.No: T7043
Synonym: 头孢替坦,Apacef
Target: Antibacterial, Antibiotic
Gemifloxacin mesylate
Cat.No: T1492
Synonym: LB-20304a,甲磺酸吉米沙星,SB-265805S,Gemifloxacin mesylate
Target: DNA gyrase, Topoisomerase, Antibacterial
Chlorhexidine digluconate
Cat.No: T14951
Synonym:
Target: Apoptosis, Antibiotic
Omeprazole Sodium
Cat.No: T22391
Synonym:
Target: P450, Proton pump, Antibacterial, Autophagy
Cefpodoxime proxetil
Cat.No: T4998
Synonym:
Target: Antibacterial, Antibiotic
Nitrofural
Cat.No: T9449
Synonym: [(E)-(5-nitrofuran-2-yl)methylideneamino,(E)-2-((5-硝基呋喃-2-基)亚甲基)肼甲酰胺
Target: Antibacterial
Secnidazole
Cat.No: T0195
Synonym: RP-14539,PM-185184,塞克硝唑
Target: Antibiotic, Parasite
Ceftezole sodium
Cat.No: T7858
Synonym: Celoslin,Falomesin,头孢替唑钠,Alomen
Target: Anti-infection, Antibacterial, Antibiotic, Glucosidase
Cefixime
Cat.No: T0932
Synonym: FK-027,头孢克肟,Cefspan,Cefiximum,Cephoral,FR-17027,CL-284635
Target: Antibacterial, Antibiotic
Flumequine
Cat.No: T1060
Synonym: Flumigal,氟甲喹,R-802
Target: Topoisomerase, Antibacterial, Antibiotic
Cefotaxime sodium
Cat.No: T0911
Synonym: Cefotaxim sodium salt,头孢噻肟钠,Cefotaxime sodium salt,Cefotaxim (sodium salt),HR-756 (sodium salt)
Target: Antibacterial, Antibiotic
Imipenem
Cat.No: T124492
Synonym: N-Formimidoyl thienamycin,MK0787
Target: Antifungal
Cat. No. Product Name Target Signaling Pathways
T2P2937 Nonacosane

Others; Antibacterial Microbiology/Virology; Others
Nonacosane 是从Baphia massaiensis 分离的,是一种由 29 个碳原子组成的直链烷烃,具有植物代谢物和挥发油成分的作用。
T8160 EGCG Octaacetate

乙酰化表没食子儿茶素没食子酸酯,乙酰化EGCG

Others; Antibacterial Microbiology/Virology; Others
EGCG Octaacetate 是表没食子儿茶素没食子酸酯的前药,对革兰氏阳性菌和革兰氏阴性菌有潜在抗菌可能。它可下调 PI3K/Akt/NFκB 磷酸化和 p65 乙酰化来降低促炎介质水平,减少小鼠结肠炎引起的结肠癌。
T0971 Dirithromycin

Dirithromycinum,地红霉素,ASE 136,LY237216,Diritromicina,Dirithromycine

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Dirithromycin (LY237216) 是一种红霉素衍生物,是一种具有口服活性的半合成大环内酯类抗生素。它用于治疗许多不同类型的细菌感染。
T10662L Calcimycin

Antibiotic A-23187,离子载体(钙镁盐混合物),A-23187

Apoptosis; Antibacterial; Antibiotic; Autophagy; Antifungal Apoptosis; Autophagy; Microbiology/Virology
Calcimycin (A-23187) 是抗生素和二价阳离子离子载体。它抑制革兰氏阳性细菌和一些真菌生长,也抑制 ATP 酶的活性并解耦哺乳动物细胞的氧化磷酸化。它通过增加细胞内钙浓度诱导 Ca2+依赖性细胞死亡。
TQ0251 (Z)-2-decenoic acid

(Z)-dec-2-enoic acid,(Z)-2-癸烯酸,cis-2-Decenoic acid,cis-dec-2-enoic acid

Others Others
(Z)-2-decenoic acid (cis-dec-2-enoic acid) 是一种由铜绿假单胞菌产生的不饱和脂肪酸。它能够诱导一系列革兰氏阴性细菌(包括铜绿假单胞菌)和革兰氏阳性细菌形成的生物膜发生分散反应。它能够抑制生物膜发育。
T8247 (+)-Aromadendrene

Anti-infection Microbiology/Virology
(+)-Aromadendrene 是一种天然产物,对革兰氏阳性菌和革兰氏阴性菌具有显着的抗菌活性。
T1665 Daptomycin

达托霉素,LY146032

DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Daptomycin (LY146032) 是脂肽类抗生素,在体外快速灭活革兰氏阳性细菌。
T8062 Cefazedone

Refosporen,头孢西酮

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Cefazedone (Refosporen) 是一种具有抗革兰氏阳性和革兰氏阴性菌活性的时间依赖性头孢菌素抗生素。
TN2279 Totarol

(+)-Totarol,桃柁酚

Antibacterial; Antifection Microbiology/Virology
Totarol ((+)-Totarol) 对几种致病性革兰氏阳性细菌、结核分枝杆菌具有抗菌作用。
T1134 Clofoctol

叔辛酚氯,氯福克酚

Antibacterial; Antibiotic Microbiology/Virology
Clofoctol 是一种抗生素,,可研究革兰氏阳性菌感染。它仅对革兰氏阳性菌起作用, 可渗透入人类肺组织。
T5037 Midecamycin

Antibiotic SF-837,Turimycin P3,Medecamycin A1,Rubimycin,麦迪霉素,Platenomycin B1,Espinomycin A

Antibacterial; Antibiotic Microbiology/Virology
Midecamycin (Medecamycin A1) 是乙酰氧基取代的大环内酯类抗生素,对革兰氏阳性和阴性菌有效。
T1306 Norfloxacin

氟哌酸,MK-0366,诺氟沙星

DNA gyrase; Topoisomerase; Endogenous Metabolite; Antibacterial; Antibiotic DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Norfloxacin (MK-0366) 是广谱抗生素,能通过结合DNA 旋转酶抑制革兰氏阳性和阴性菌。
T1679 Thiostrepton

Thiactin,Bryamycin,Alaninamide,硫链丝菌素

DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Thiostrepton (Alaninamide) 是一种选择性抑制FOXM1的抗生素。FOXM1会与 YAP/TEAD 复合物结合,形成YAP/TEAD/FOXM1 复合物。
T8302 Ceftiofur

Antibacterial; Antibiotic Microbiology/Virology
Ceftiofur 是一种半合成抗生素,对家畜的各种革兰氏阳性和革兰氏阴性菌、好氧菌和厌氧菌均有抗菌活性。
T0814L Ampicillin

Amcill,D-(-)-α-Aminobenzylpenicillin,Aminobenzylpenicillin,氨苄青霉素,Ampicillin acid

Antibacterial; Antibiotic Microbiology/Virology
Ampicillin (Aminobenzylpenicillin) 属于 β-内酰胺类抗生素,是一种半合成的青霉素。Ampicillin 具有杀菌活性,对各种革兰氏阳性细菌和革兰氏阴性细菌均有抑制活性。
T5S0814 Berberine hydrogen sulphate

Berberine Bisulfate,硫酸氢黄连素,Umbellatine Sulfate

Antibacterial Microbiology/Virology
Berberine hydrogen sulphate (Umbellatine Sulfate) 是一种从几种植物中提取的生物碱,对多种微生物具有抗菌活性,包括革兰氏阳性和革兰氏阴性细菌、真菌和原生动物。
T5274 D-​(+)​-​Phenyllactic acid

D-3-苯乳酸,D-3-Phenyllactic acid

Endogenous Metabolite; Antibacterial Metabolism; Microbiology/Virology
D-​(+)​-​Phenyllactic acid (D-3-Phenyllactic acid) 是一种由白地霉分泌得到的抗菌剂,可抑制部分来自人类和食品的革兰氏阳性菌以及来自人类的革兰氏阴性菌。
T8504 Dianemycin

Nanchangmycin (free acid)

Antibacterial; Antibiotic Microbiology/Virology
Dianemycin (Nanchangmycin (free acid)) 由Streptomyces nanchangensis 产生的一种聚醚抗生素,抑制革兰氏阳性菌。它也是一种针对 Zika 病毒的广谱抗病毒药物。
T5003 Rifamycin sodium

Rifamycin sodium salt,利福霉素钠

Antibacterial; Antibiotic Microbiology/Virology
Rifamycin sodium (Rifamycin sodium salt) salt 是从地中海曲霉或其突变体的发酵中分离出来的一种安沙霉素抗生素家族。它对革兰氏阳性菌和某些革兰氏阴性菌有抗生素活性。
TN1651 Furanodiene

Apoptosis; PARP; Reactive Oxygen Species; Caspase; CDK; P-gp Apoptosis; Cell Cycle/Checkpoint; Chromatin/Epigenetic; DNA Damage/DNA Repair; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience; NF-κB; Proteases/Proteasome
Furanodiene 是从姜黄中提取的一种萜类天然产物,可抑制外排转运蛋白Pgp 功能并降低 Pgp 蛋白水平。它通过抗血管生成和诱导ROS 产生,DNA 链断裂和细胞凋亡发挥抗癌作用。
T0906 Salinomycin

盐霉素,Procoxacin

Wnt/beta-catenin; Antibacterial Cytoskeletal Signaling; Microbiology/Virology; Stem Cells
Salinomycin (Procoxacin)是一种多醚类钾离子载体抗生素,特异性抑制革兰氏阳性细菌生长。Salinomycin 作为Wnt/β-连环蛋白信号通路的有效抑制剂,阻断Wnt诱导的LRP6磷酸化。此外,Salinomycin (Procoxacin)对人类癌症干细胞显示出选择性活性。
T0958 Penicillin G sodium salt

青霉素钠,Penicillin G Sodium,Benzylpenicillin sodium salt,Benzylpenicillin Sodium

GABA Receptor; Antibacterial; Antibiotic Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience
Penicillin G sodium(Benzylpenicillin sodium) salt 是一种 β-内酰胺类抗生素。
T12830 Sapienic acid sodium

Antibacterial Microbiology/Virology
Sapienic acid sodium,主要存在于皮肤和粘膜中的脂肪酸,对皮肤和口腔内的革兰氏阳性及阴性细菌展现出不同程度的抗菌效果。其对血链球菌、微生物链球菌与核纤梭菌的抗菌活性表现,MBC值分别为31.3 μg/mL、375.0 μg/mL与93.8 μg/mL。
T20643 Cefoxitin

Rephoxitin,Cefoxitinum

Cell wall; Antibacterial; Antibiotic Immunology/Inflammation; Microbiology/Virology
Cefoxitin (Rephoxitin) 是一种广谱的、可口服的第二代头孢霉素类抗生素。Cefoxitin 干扰细菌细胞壁的合成。其活性谱包括革兰氏阴性和革兰氏阳性菌,通常用于腹腔感染、盆腔感染和某些类型的妇科感染等腹部,对厌氧菌具有高效性。
TN7231 Di-O-methylhonokiol

Honokiol dimethyl ether

Antioxidant oxidation-reduction
Di-O-methylhonokiol (Honokiol dimethyl ether) 是Magnolia grandiflora L 的酚类成分,具有抗微生物活性,对革兰氏阳性和抗酸细菌和真菌具有显著的抗氧化活性。
T2989 4-Hydroxybenzoic acid

p-hydroxybenzoic acid,para-Hydroxybenzoic acid,PHBA,对羟基苯甲酸,4-hydroxybenzoate

Endogenous Metabolite; Antibacterial Metabolism; Microbiology/Virology
4-Hydroxybenzoic acid (4-hydroxybenzoate) 是苯甲酸的酚衍生物,可抑制革兰氏阳性和革兰氏阴性菌,IC50值为160 μg/mL。
T4S0867 Pogostone

DHELWANGIN,广藿香酮

Apoptosis; Antibacterial; Autophagy Apoptosis; Autophagy; Microbiology/Virology
Pogostone (DHELWANGIN) 是从薄荷中分离出,对革兰氏阴性菌、革兰氏阳性菌、大肠埃希菌等具有强效抗菌、抗真菌活性。它诱导细胞凋亡和自噬。
T8347 Rifamycin S

Reactive Oxygen Species; ROS; Antibacterial; Antibiotic Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
Rifamycin S 是一种 DNA 依赖性 RNA 聚合酶抑制剂,是一种醌和一种针对革兰氏阳性细菌的抗生素试剂。它是涉及两个电子的可逆氧化还原系统的氧化形式。它能产生活性氧并抑制微粒体脂质过氧化,可研究肺结核和麻风病。
T1219 Sisomicin Sulfate

硫酸西索米星,Pathomycin,Extramycin,硫酸西索紫苏

Antibacterial; Antibiotic Microbiology/Virology
Sisomicin Sulfate (Pathomycin) 是由Micromonospora inyoensis 产生的一种广谱氨基糖苷类抗生素,对革兰氏阳性细菌有很大活性。
T3092 Nigericin sodium salt

尼日利亚菌素,尼日利亚菌素钠盐

Potassium Channel; NOD-like Receptor (NLR); Antibacterial; Antibiotic; NOD Immunology/Inflammation; Membrane transporter/Ion channel; Microbiology/Virology; NF-κB
Nigericin sodium salt 属于抗生素,是一种 NLRP3 激活剂,也是一种阳离子离子载体。Nigericin sodium 可以触发 NALP3 炎性体的激活,可抑制高尔基体功能并抑制革兰氏阳性菌的生长。
T0819 Spiramycin

Espiramicin,螺旋霉素,Sequamycin,Rovamycin,Provamycin,Formacidine

Antibacterial; Antibiotic; Parasite Microbiology/Virology
Spiramycin (Rovamycin) 是一种由安博链霉菌产生的大环内酯类抗生素,具有抗细菌和弓形虫活性,并具有抗寄生虫作用。它由 16 个内酯环组成,其上附着 mycaminose,forosamine 和 mycarose 三种糖。
T4S1943 Kirenol

奇壬醇,奇任醇,Kirel

Wnt/beta-catenin Cytoskeletal Signaling; Stem Cells
Kirenol (Kirel) 是分离自 Siegesbeckia orientalis 中的,具有抗氧化、抗炎、抗过敏、抗关节炎活性,可用于缓解疼痛的研究。
T26805 Bicyclomycin

Bicozamycin

Bicyclomycin is a broad spectrum antibiotic active against Gram-negative bacteria and the Gram-positive bacterium, Micrococcus luteusn.
TN4518 Meridinol

Antifection Microbiology/Virology
Meridinol has wide antimicrobial activity, includes against gram-positive and gram-negative bacteria and fungi.
T11551 Helvolic acid

Fumigacin

Others Others
Helvolic acid, an antibiotic derived from Xylaria sp., exhibits effectiveness against Gram-positive bacteria.
TN6002 Crenatine

1-Ethyl-4-methoxy-β-carboline

Crenatine possesses antibacterial activity, it is more effective against Gram-positive than Gram-negative bacteria.
T27024 Citromycetin

Frequentic Acid,NSC-53584,NSC 53584,NSC53584

Citromycetin is a fungal metabolite originally isolated from Australian P. frequentans. It has antibiotic activity against the Gram-negative bacteria V. cholerae and S. flexneri and the Gram-positive bacteria S. aureus.
T38176 Muramic acid

Muramic acid is a prevalent constituent found in the cell walls of Gram-positive bacteria, serving as a distinguishing marker for such bacteria[1].
TN1301 6,8-Diprenylgenistein

6,8-二异戊烯基金雀异黄素,鲁冰花

Antifection Microbiology/Virology
6,8-Diprenylgenistein has antimicrobial activity, it has anti-bacteria activity against Gram-negative and Gram-positive bacteria.
T4131 Arjunic acid

COX; Antifection Immunology/Inflammation; Microbiology/Virology; Neuroscience
Arjunic acid is a strong antioxidant and a free radical scavenger. Arjunic acid shows activity against Gram-positive and Gram-negative bacteria with MIC values ranging between 1.9 and 15.6 microg/mL.
TN6163 3-O-cis-p-Coumaroylmaslinic acid

3-beta-O-(trans-p-Coumaroyl)maslinic acid shows antimicrobial activity on Gram-positive bacteria and yeasts.
TN2502 1,5,6-Trihydroxyxanthone

Others Others
1,5,6-Trihydroxyxanthone exhibits antibacterial activity against Gram-positive bacteria.
TN4264 Isoapetalic acid

胡桐,海棠木

HIV Protease; Antifection Microbiology/Virology; Proteases/Proteasome
Isoapetalic acid and apetalic acid exhibit cytotoxic activities towards both cancer cell lines(human breast cancer (MCF-7) and human lung carcinoma (A-549) cell lines) and both Gram-positive bacteria(two Gram-positive bacteria, S. aureus and B. subtilis a
T16673 Pseudouridimycin

PUM

Others Others
Pseudouridimycin is a C-nucleoside analogue. Pseudouridimycin is an antibiotic and is a selective bacterial RNA polymerase (RNAP) inhibitor. It is effective against both Gram-negative and Gram-positive bacteria.
TN6148 3-O-trans-p-Coumaroylmaslinic acid

3-beta-O-(trans-p-Coumaroyl)maslinic acid is a DNA polymerase B" inhibitor. It shows antimicrobial activity on Gram-positive bacteria and yeasts.
TN5930 Ocotillone

Ocotillone has potent antibacterial activity against Gram-negative bacteria, P. aeruginosa and S. typhimurium, that are without hemolytic activity, whereas it has weak antimicrobial activity against Gram-positive bacteria and fungi. Ocotillone shows only
T32924 Lucidin ethyl ether

Ibericin 是一种从Prismatomeris filamentosa 根中分离得到的蒽醌代谢产物,对革兰氏阳性菌和革兰氏阴性菌具有一定的抗菌活性。
T71909 Kumbicin C

Kumbicin C inhibits the growth of NS-1 mouse myeloma cells (IC50 = 0.74 μg/ml) and the growth of the Gram-positive bacteria B. subtilis (MIC = 1.6 μg/ml).
T10455 Bafilomycin B1

巴佛洛霉素 B1

Others Others
Bafilomycin B1, a macrolide antibiotic isolated from Streptomyces sp, acts as an inhibitor of K+-dependent ATPase of E. coli. It also inhibits Gram-positive bacteria and fungi.
T27977 Manzamine A

Keramamine A

Manzamine A is a GSK-3 inhibitor and vacuolar ATPase uncoupler found in marine sponges. It inhibits autophagy and tumor growth in cancer models, suppresses foam cell formation in macrophages, prevents growth of gram negative and gram positive bacteria, an
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天然产物

Nonacosane
Cat.No: T2P2937
Synonym:
Target: Others, Antibacterial
EGCG Octaacetate
Cat.No: T8160
Synonym: 乙酰化表没食子儿茶素没食子酸酯,乙酰化EGCG
Target: Others, Antibacterial
Dirithromycin
Cat.No: T0971
Synonym: Dirithromycinum,地红霉素,ASE 136,LY237216,Diritromicina,Dirithromycine
Target: ribosome, Antibacterial, Antibiotic
Calcimycin
Cat.No: T10662L
Synonym: Antibiotic A-23187,离子载体(钙镁盐混合物),A-23187
Target: Apoptosis, Antibacterial, Antibiotic, Autophagy, Antifungal
(Z)-2-decenoic acid
Cat.No: TQ0251
Synonym: (Z)-dec-2-enoic acid,(Z)-2-癸烯酸,cis-2-Decenoic acid,cis-dec-2-enoic acid
Target: Others
(+)-Aromadendrene
Cat.No: T8247
Synonym:
Target: Anti-infection
Daptomycin
Cat.No: T1665
Synonym: 达托霉素,LY146032
Target: DNA/RNA Synthesis, Antibacterial, Antibiotic
Cefazedone
Cat.No: T8062
Synonym: Refosporen,头孢西酮
Target: Others, Antibacterial, Antibiotic
Totarol
Cat.No: TN2279
Synonym: (+)-Totarol,桃柁酚
Target: Antibacterial, Antifection
Clofoctol
Cat.No: T1134
Synonym: 叔辛酚氯,氯福克酚
Target: Antibacterial, Antibiotic
Midecamycin
Cat.No: T5037
Synonym: Antibiotic SF-837,Turimycin P3,Medecamycin A1,Rubimycin,麦迪霉素,Platenomycin B1,Espinomycin A
Target: Antibacterial, Antibiotic
Norfloxacin
Cat.No: T1306
Synonym: 氟哌酸,MK-0366,诺氟沙星
Target: DNA gyrase, Topoisomerase, Endogenous Metabolite, Antibacterial, Antibiotic
Thiostrepton
Cat.No: T1679
Synonym: Thiactin,Bryamycin,Alaninamide,硫链丝菌素
Target: DNA/RNA Synthesis, Antibacterial, Antibiotic
Ceftiofur
Cat.No: T8302
Synonym:
Target: Antibacterial, Antibiotic
Ampicillin
Cat.No: T0814L
Synonym: Amcill,D-(-)-α-Aminobenzylpenicillin,Aminobenzylpenicillin,氨苄青霉素,Ampicillin acid
Target: Antibacterial, Antibiotic
Berberine hydrogen sulphate
Cat.No: T5S0814
Synonym: Berberine Bisulfate,硫酸氢黄连素,Umbellatine Sulfate
Target: Antibacterial
D-​(+)​-​Phenyllactic acid
Cat.No: T5274
Synonym: D-3-苯乳酸,D-3-Phenyllactic acid
Target: Endogenous Metabolite, Antibacterial
Dianemycin
Cat.No: T8504
Synonym: Nanchangmycin (free acid)
Target: Antibacterial, Antibiotic
Rifamycin sodium
Cat.No: T5003
Synonym: Rifamycin sodium salt,利福霉素钠
Target: Antibacterial, Antibiotic
Furanodiene
Cat.No: TN1651
Synonym:
Target: Apoptosis, PARP, Reactive Oxygen Species, Caspase, CDK, P-gp
Salinomycin
Cat.No: T0906
Synonym: 盐霉素,Procoxacin
Target: Wnt/beta-catenin, Antibacterial
Penicillin G sodium salt
Cat.No: T0958
Synonym: 青霉素钠,Penicillin G Sodium,Benzylpenicillin sodium salt,Benzylpenicillin Sodium
Target: GABA Receptor, Antibacterial, Antibiotic
Sapienic acid sodium
Cat.No: T12830
Synonym:
Target: Antibacterial
Cefoxitin
Cat.No: T20643
Synonym: Rephoxitin,Cefoxitinum
Target: Cell wall, Antibacterial, Antibiotic
Di-O-methylhonokiol
Cat.No: TN7231
Synonym: Honokiol dimethyl ether
Target: Antioxidant
4-Hydroxybenzoic acid
Cat.No: T2989
Synonym: p-hydroxybenzoic acid,para-Hydroxybenzoic acid,PHBA,对羟基苯甲酸,4-hydroxybenzoate
Target: Endogenous Metabolite, Antibacterial
Pogostone
Cat.No: T4S0867
Synonym: DHELWANGIN,广藿香酮
Target: Apoptosis, Antibacterial, Autophagy
Rifamycin S
Cat.No: T8347
Synonym:
Target: Reactive Oxygen Species, ROS, Antibacterial, Antibiotic
Sisomicin Sulfate
Cat.No: T1219
Synonym: 硫酸西索米星,Pathomycin,Extramycin,硫酸西索紫苏
Target: Antibacterial, Antibiotic
Nigericin sodium salt
Cat.No: T3092
Synonym: 尼日利亚菌素,尼日利亚菌素钠盐
Target: Potassium Channel, NOD-like Receptor (NLR), Antibacterial, Antibiotic, NOD
Spiramycin
Cat.No: T0819
Synonym: Espiramicin,螺旋霉素,Sequamycin,Rovamycin,Provamycin,Formacidine
Target: Antibacterial, Antibiotic, Parasite
Kirenol
Cat.No: T4S1943
Synonym: 奇壬醇,奇任醇,Kirel
Target: Wnt/beta-catenin
Bicyclomycin
Cat.No: T26805
Synonym: Bicozamycin
Target:
Meridinol
Cat.No: TN4518
Synonym:
Target: Antifection
Helvolic acid
Cat.No: T11551
Synonym: Fumigacin
Target: Others
Crenatine
Cat.No: TN6002
Synonym: 1-Ethyl-4-methoxy-β-carboline
Target:
Citromycetin
Cat.No: T27024
Synonym: Frequentic Acid,NSC-53584,NSC 53584,NSC53584
Target:
Muramic acid
Cat.No: T38176
Synonym:
Target:
6,8-Diprenylgenistein
Cat.No: TN1301
Synonym: 6,8-二异戊烯基金雀异黄素,鲁冰花
Target: Antifection
Arjunic acid
Cat.No: T4131
Synonym:
Target: COX, Antifection
3-O-cis-p-Coumaroylmaslinic acid
Cat.No: TN6163
Synonym:
Target:
1,5,6-Trihydroxyxanthone
Cat.No: TN2502
Synonym:
Target: Others
Isoapetalic acid
Cat.No: TN4264
Synonym: 胡桐,海棠木
Target: HIV Protease, Antifection
Pseudouridimycin
Cat.No: T16673
Synonym: PUM
Target: Others
3-O-trans-p-Coumaroylmaslinic acid
Cat.No: TN6148
Synonym:
Target:
Ocotillone
Cat.No: TN5930
Synonym:
Target:
Lucidin ethyl ether
Cat.No: T32924
Synonym:
Target:
Kumbicin C
Cat.No: T71909
Synonym:
Target:
Bafilomycin B1
Cat.No: T10455
Synonym: 巴佛洛霉素 B1
Target: Others
Manzamine A
Cat.No: T27977
Synonym: Keramamine A
Target:
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