247
85
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T14391 |
Azidamfenicol
|
Antibacterial; Antibiotic | Microbiology/Virology |
Azidamfenicol 抑制核糖体肽基转移酶,Ki 为 22 µM。Azidamfenicol 是一种广谱氯霉素类抗生素。 | |||
T4998L |
Cefpodoxime (free acid)
|
Others | Others |
Cefpodoxime (free acid) 是一种口服的第三代头孢菌素抗生素。除铜绿假单胞菌、肠球菌和脆弱拟杆菌外,它对大多数革兰氏阳性和革兰氏阴性微生物均有效。 | |||
T9680 |
Irloxacin
|
Antibacterial | Microbiology/Virology |
Irloxacin 是一种口服活性的喹诺酮类抗菌剂,在酸性条件下具有更强大的活性。在体外,Irloxacin 对革兰氏阳性菌和革兰氏阴性菌都具有良好的抗菌谱。 | |||
T20525 |
Chloramphenicol palmitate
|
Antibacterial; Antibiotic | Microbiology/Virology |
Chloramphenicol palmitate 是一种广谱抗生素,对革兰氏阳性和革兰氏阴性细菌具有活性。 Chloramphenicol palmitate 可用于在含有氯霉素抗性基因的转化细胞中作为细菌选择剂的研究。 | |||
T1008 |
Cephalexin
头孢氨苄,Cefalexin,Cephacillin |
Antibacterial; Antibiotic | Microbiology/Virology |
Cephalexin (Cephacillin) 是一种强口服活性的头孢菌素抗生素。它通过破坏细菌细胞壁的生长来杀死革兰氏阳性和一些革兰氏阴性细菌。它可研究肺炎、链球菌性咽喉炎、细菌性心内膜炎等。 | |||
T5006 |
Flucloxacillin sodium
氟氯西林钠,floxacillin sodium |
Antibacterial; Antibiotic | Microbiology/Virology |
Flucloxacillin sodium (floxacillin sodium) 是一种高活性抗生素,抑制革兰氏阳性和革兰氏阴性菌。 | |||
T6582 |
Mezlocillin Sodium
美洛西林钠,Baycipen |
Antibacterial; Antibiotic | Microbiology/Virology |
Mezlocillin Sodium (Baycipen) 是一种青霉素 β-内酰胺类抗生素,用于治疗由易感染微生物引起的细菌感染。 | |||
T3117 |
Marbofloxacin
马波沙星,Marbofloxacine,Zeniquin,Marbocyl |
Topoisomerase; Antibacterial; Antibiotic | DNA Damage/DNA Repair; Microbiology/Virology |
Marbofloxacin (Zeniquin) 是一种具有口服活性的氟喹诺酮类广谱抗菌剂。它可研究革兰氏阳性和革兰氏阴性细菌以及支原体引起的感染。 | |||
TP1444 |
Magainin 2
蛙皮素 2 |
Antibacterial; Antibiotic; Antifungal | Microbiology/Virology |
Magainin 2是从非洲爪蟾皮肤中分离得到的一种抗菌肽。它对许多革兰氏阴性和革兰氏阳性细菌显示出抗生素活性,对原生动物也有活性。它通过优先与细菌膜中丰富的阴离子磷脂相互作用而发挥细胞毒性作用。 | |||
T0396 |
Pipemidic acid
吡哌酸,Acido pipemidico |
Antibacterial; Antibiotic | Microbiology/Virology |
Pipemidic acid (Acido pipemidico) 是一种新型抗菌剂,对革兰氏阴性菌和某些革兰氏阳性细菌具有活性,可研究肠道、泌尿和胆道感染。 | |||
T0116 |
Balofloxacin
|
DNA gyrase; Antibacterial; Antibiotic | DNA Damage/DNA Repair; Microbiology/Virology |
Balofloxacin 是一种具有口服活性的氟喹诺酮类抗生素,可通过干扰 DNA 促旋酶来抑制细菌 DNA 的合成,对革兰氏阴性,革兰氏阳性和厌氧菌具有广谱抗菌活性。它可研究呼吸道,肠道和泌尿道感染。 | |||
T9066 |
Merafloxacin
CI 934 |
SARS-CoV | Microbiology/Virology |
Merafloxacin (CI 934) 是一种氟喹诺酮类抗菌药物,也被确定为 SARS-CoV-2 的 1 PRF 抑制剂。它对革兰氏阳性菌和革兰氏阴性菌具有体外活性。 | |||
T7865 |
Danofloxacin
达氟沙星,达诺沙星,Danofloxacino,Danofloxacin free base,Danofloxacine |
Others; DNA/RNA Synthesis; Antibacterial; Antibiotic | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others |
Danofloxacin (Danofloxacin free base) free base 是一种具有口服活性第三代氟喹诺酮抗菌剂,对大多数革兰氏阴性和革兰氏阳性细菌,支原体和衣原体物种具有广谱的活性,并通过抑制细菌的 DNA 回转酶发挥抗菌作用。它可用于牛,猪和鸡呼吸道疾病的研究。 | |||
T2692 |
A40926
Dalbavancin Impurity,达巴霉素杂质 |
Antibacterial | Microbiology/Virology |
A40926 (Dalbavancin Impurity) 是Dalbavancin 的前体,是一种糖肽抗生素。它抑制革兰氏阳性细菌,对淋病奈瑟氏球菌非常有效。 | |||
T0133 |
Cefdinir
FK-482,头孢地尼,CI-983,PD 134393 |
Glutathione Peroxidase; Antibacterial; Antibiotic | Metabolism; Microbiology/Virology |
Cefdinir (FK-482) 是头孢菌素类中的一种半合成广谱抗生素,对几种革兰氏阴性和革兰氏阳性细菌引起的感染有效。它可研究耳,鼻窦,喉咙和皮肤的常见细菌感染。 | |||
T73997 | Anti gram-positive/negative bacteria agent 1 | ||
Anti gram-positive/negative bacteria agent 1 是一种含有基于MECAM的人工铁载体的抗生素化合物。 | |||
T20774 |
Sarafloxacin
A-56620,A 56620,A56620,沙拉沙星 |
Antibacterial; Antibiotic | Microbiology/Virology |
Sarafloxacin (A56620) 对革兰氏阳性菌和革兰氏阴性菌具有抗菌活性。 | |||
T1640 |
Ciprofloxacin
Ciproxan,环丙沙星,Ciprobay,Bay o 9867,Bay-09867 |
Topoisomerase; Antibacterial; Antibiotic | DNA Damage/DNA Repair; Microbiology/Virology |
Ciprofloxacin (Bay-09867) 是一种有高抗菌活性的氟喹诺酮类抗生素。 | |||
T11315 |
Fosmidomycin sodium salt
FR-31564 sodium salt |
Antibiotic; Parasite | Microbiology/Virology |
Fosmidomycin sodium salt (FR-31564 sodium salt) 是一种抗感染类抗生素,具有抗疟疾活性,抑制革兰氏阴性菌和革兰氏阳性菌。 | |||
T11301L |
Flomoxef sodium
|
Others | Others |
Flomoxef sodium 属于奥沙环类抗生素,对多种革兰氏阳性菌均具有良好的杀灭活性。 | |||
T0425 |
Pefloxacin Mesylate
Pefloxacinium mesylate,甲磺酸培氟沙星 |
Topoisomerase; Antibacterial; Antibiotic | DNA Damage/DNA Repair; Microbiology/Virology |
Pefloxacin Mesylate (Pefloxacinium mesylate) 是一种抗菌化合物,可抑制DNA 旋转酶阻断DNA 复制。 | |||
T11123 |
DuP 105
|
Antibacterial; Antibiotic | Microbiology/Virology |
DuP 105是可口服的oxazolidinone类化合物,这是一种新型合成的抗菌化合物,对革兰氏阳性细菌具有有效性。 | |||
T6706 |
Ticarcillin sodium
Ticarpen hydrate,Aerugipen hydrate,替卡西林单钠盐单水合物,BRL 2288,AB 2288,Monapen |
Others; Antibacterial; Antibiotic | Microbiology/Virology; Others |
Ticarcillin sodium (Aerugipen hydrate) 主要用于抗革兰氏阴性菌, 也能用于研究嗜麦芽感染。 | |||
TP1763L |
Magainin 1 acetate
|
Antibacterial; Antibiotic; Antifungal | Microbiology/Virology |
Magainin 1 acetate 是一种抗菌肽。它对许多革兰氏阴性和革兰氏阳性细菌表现出抗生素活性。 | |||
T4020 |
Cadazolid
ACT-179811,卡达唑利德 |
Antibacterial; Antibiotic | Microbiology/Virology |
Cadazolid (ACT-179811) 是一种新型恶唑烷酮类抗生素,对Clostridium difficile 有活性。 | |||
T73054 |
Moiramide B
|
Acetyl-CoA Carboxylase; Antibiotic | Metabolism; Microbiology/Virology |
Moiramide B 是一种高效的乙酰辅酶 A 羧化酶 (ACC) 抑制剂(IC50:6 nM),具有抗菌活性,强烈抑制革兰氏阳性菌,但对革兰氏阴性菌的抑制效果较弱。 | |||
TP1663L |
CysHHC10 acetate
CysHHC10 acetate(1408311-03-4 free base) |
Antibacterial | Microbiology/Virology |
CysHHC10 acetate 对革兰氏阳性菌和革兰氏阴性菌均具有抗菌活性,对大肠杆菌、铜绿假单胞菌、金黄色葡萄球菌和表皮葡萄球菌的 MIC 分别为 10.1、20.2、2.5 和 1.3 mM。 | |||
T28229 |
Olanexidine hydrochloride
OPB2045,OPB-2045,OPB-2045 HCl,OPB 2045 |
Antibacterial | Microbiology/Virology |
Olanexidine hydrochloride (OPB-2045 HCl) 对革兰氏阳性菌和革兰氏阴性菌具有杀菌活性。 Olanexidine hydrochloride 破坏金黄色葡萄球菌的膜完整性。 | |||
T0967 |
Teicoplanin
Antibiotic MDL-507,MDL-507,替考拉宁,Teichomycin |
Antibacterial; Antibiotic | Microbiology/Virology |
Teicoplanin (MDL-507) 是一种半合成的糖肽抗生素, 可用于由革兰氏阳性菌引起的严重感染的相关研究。 | |||
T22228 |
Tylvalosin tartrate
酒石酸乙酰异戊酰泰乐菌素,Acetylisovaleryltylosin Tartrate |
Antibacterial; Antibiotic | Microbiology/Virology |
Tylvalosin tartrate (Acetylisovaleryltylosin Tartrate) 是一种对革兰氏阳性细菌具有抗性的大环内酯类抗生素。 | |||
T17021 |
Tebipenem
LJC 11036 |
Antibiotic | Microbiology/Virology |
Tebipenem 是一种口服碳青霉烯类抗生素。 它对革兰氏阳性和阴性细菌具有广谱活性。 | |||
T3247 |
Lysozyme from chicken egg white
鸡蛋清溶菌酶,溶菌酶,Lysozyme |
Others; Antibacterial | Microbiology/Virology; Others |
Lysozyme from chicken egg white (Lysozyme) 是一种存在于鸡蛋清中的杀菌酶,它溶解革兰氏阳性菌。 | |||
T0897 |
Nitrofurazone
NFZ,呋喃西林,Nitrofural,Furacilin |
Dehydrogenase; Antibacterial; Glutathione reductase; Antibiotic | Metabolism; Microbiology/Virology; oxidation-reduction |
Nitrofurazone (Furacilin) 是一种抗生素。 | |||
T19709 |
Nitrocefin
|
Others | Others |
Nitrocefin 是 β-内酰胺酶的显色底物,当 β-内酰胺酶将 β-内酰胺环中的酰胺键水解后,Nitrocefin 的颜色会由黄色变为红色。它可用于 β-内酰胺酶耐药抗生素的研究。 | |||
T19860 |
Clavulanic Acid
BRL 14151,MM-14151,MM 14151,RX-10100,MM14151,BRL14151,BRL-14151 |
Antibacterial; Antifungal | Microbiology/Virology |
Clavulanic Acid(RX-10100) 是一种由生物体克拉维链霉菌产生的主要β-内酰胺类抗生素,是一种强效的细菌 β-内酰胺酶抑制剂,用于研究细菌引起的感染。Clavulanic Acid 具有广谱的生物活性,对多种革兰氏阳性和革兰氏阴性细菌均有活性。 | |||
T1001 |
Dicloxacillin Sodium hydrate
Dicloxacillin sodium salt monohydrate,双氯西林钠,Dicloxacillin sodium monohydrate |
Antibacterial; Antibiotic | Microbiology/Virology |
Dicloxacillin Sodium hydrate 是一种青霉素类窄谱β内酰胺抗生素,可研究革兰氏阳性菌感染。 | |||
T22408 |
Proflavine
吡啶-3,6-二胺,3,6-Diaminoacridine |
Antibacterial | Microbiology/Virology |
Proflavine (3,6-Diaminoacridine) 是吖啶染料,可用作抗菌剂。它是 DNA 嵌入剂,能够阻滞Kir3.2孔。它用作与 Kir3.2 相关的神经系统疾病的研究。 | |||
T68137 |
Sanfetrinem
GV104326 |
Antibiotic | Microbiology/Virology |
Sanfetrinem (GV104326) sodium 是一种新型可口服 β-内酰胺酶抗生素,对革兰氏阳性菌和革兰氏阴性菌显示出显著的抗菌活性,可用于研究细菌感染。 | |||
T7043 |
Cefotetan
头孢替坦,Apacef |
Antibacterial; Antibiotic | Microbiology/Virology |
Cefotetan (Apacef) 是一种半合成的头霉素抗生素,能抑制细胞壁合成发挥杀菌作用。 | |||
T1492 |
Gemifloxacin mesylate
LB-20304a,甲磺酸吉米沙星,SB-265805S,Gemifloxacin mesylate |
DNA gyrase; Topoisomerase; Antibacterial | DNA Damage/DNA Repair; Microbiology/Virology |
Gemifloxacin mesylate (Gemifloxacin mesylate) 是一种喹诺酮类口服广谱抗菌剂,可研究轻中度肺炎和慢性支气管炎的急性细菌性发作。 | |||
T14951 | Chlorhexidine digluconate | Apoptosis; Antibiotic | Apoptosis; Microbiology/Virology |
Chlorhexidine digluconate 是一种广谱防腐剂和消毒剂,具有广谱抗菌活性,抑制革兰氏阳性菌和革兰氏阴性菌,可诱导细胞坏死和凋亡,可用于研究细菌感染。 | |||
T22391 |
Omeprazole Sodium
|
P450; Proton pump; Antibacterial; Autophagy | Autophagy; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology |
Omeprazole 是有效的质子泵抑制剂,在胃肠道疾病的研究中具有价值。它竞争性抑制CYP2C19活性,Ki 为 2 到 6 μM。它还抑制革兰氏阴性菌和革兰氏阳性菌生长。它是中性鞘磷脂酶的外泌体抑制剂。 | |||
T4998 |
Cefpodoxime proxetil
|
Antibacterial; Antibiotic | Microbiology/Virology |
Cefpodoxime Proxetil 是一种口服的广谱型抗生素。它与青霉素结合蛋白结合,抑制肽聚糖的合成,干扰细菌细胞壁的生物合成。 | |||
T9449 |
Nitrofural
[(E)-(5-nitrofuran-2-yl)methylideneamino,(E)-2-((5-硝基呋喃-2-基)亚甲基)肼甲酰胺 |
Antibacterial | Microbiology/Virology |
Nitrofural 是 20 世纪已在临床应用中确立的硝基呋喃。 Nitrofural 在临床上对广泛的革兰氏阳性和革兰氏阴性细菌(包括许多常见的泌尿道病原体菌株)仍然有效。 | |||
T0195 |
Secnidazole
RP-14539,PM-185184,塞克硝唑 |
Antibiotic; Parasite | Microbiology/Virology |
Secnidazole (PM-185184) 是一种具有口服活性唑类抗生素,半衰期比甲硝唑更长。它有潜力研究细菌性阴道病。 | |||
T7858 |
Ceftezole sodium
Celoslin,Falomesin,头孢替唑钠,Alomen |
Anti-infection; Antibacterial; Antibiotic; Glucosidase | Metabolism; Microbiology/Virology |
Ceftezole sodium (Falomesin) 是一种广谱 cephem 抗生素,具有抑制多种革兰氏阳性菌和革兰氏阴性菌活性。它是一种α-葡萄糖苷酶抑制剂,具有体内抗糖尿病活性。 | |||
T0932 |
Cefixime
FK-027,头孢克肟,Cefspan,Cefiximum,Cephoral,FR-17027,CL-284635 |
Antibacterial; Antibiotic | Microbiology/Virology |
Cefixime (FR-17027) 是一种头孢菌素类抗生素, 可研究一些细菌感染。 | |||
T1060 |
Flumequine
Flumigal,氟甲喹,R-802 |
Topoisomerase; Antibacterial; Antibiotic | DNA Damage/DNA Repair; Microbiology/Virology |
Flumequine (R-802) 是一种喹诺酮类抗生素,对革兰氏阳性菌和革兰氏阴性菌均有效。它是拓扑异构酶 II 抑制剂, 抑制细胞分裂,IC50值为 15 μM (3.92 μg/mL)。 | |||
T0911 |
Cefotaxime sodium
Cefotaxim sodium salt,头孢噻肟钠,Cefotaxime sodium salt,Cefotaxim (sodium salt),HR-756 (sodium salt) |
Antibacterial; Antibiotic | Microbiology/Virology |
Cefotaxime sodium (Cefotaxim sodium salt) 是头孢类抗生素和耐内酰胺酶的头孢菌素,有抗革兰氏阳性菌和革兰氏阴性菌作用。 | |||
T124492 |
Imipenem
N-Formimidoyl thienamycin,MK0787 |
Antifungal | Microbiology/Virology |
Imipenem (MK0787) 是一种噻吩霉素衍生物,属于抗生素类,具有抗菌活性,对革兰氏阳性和革兰氏阴性菌具有部分的抑制作用。Imipenem 可用于研究碳青霉烯类非易感性感染和铜绿假单胞菌生物膜感染。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2P2937 |
Nonacosane
|
Others; Antibacterial | Microbiology/Virology; Others |
Nonacosane 是从Baphia massaiensis 分离的,是一种由 29 个碳原子组成的直链烷烃,具有植物代谢物和挥发油成分的作用。 | |||
T8160 |
EGCG Octaacetate
乙酰化表没食子儿茶素没食子酸酯,乙酰化EGCG |
Others; Antibacterial | Microbiology/Virology; Others |
EGCG Octaacetate 是表没食子儿茶素没食子酸酯的前药,对革兰氏阳性菌和革兰氏阴性菌有潜在抗菌可能。它可下调 PI3K/Akt/NFκB 磷酸化和 p65 乙酰化来降低促炎介质水平,减少小鼠结肠炎引起的结肠癌。 | |||
T0971 |
Dirithromycin
Dirithromycinum,地红霉素,ASE 136,LY237216,Diritromicina,Dirithromycine |
ribosome; Antibacterial; Antibiotic | Microbiology/Virology |
Dirithromycin (LY237216) 是一种红霉素衍生物,是一种具有口服活性的半合成大环内酯类抗生素。它用于治疗许多不同类型的细菌感染。 | |||
T10662L |
Calcimycin
Antibiotic A-23187,离子载体(钙镁盐混合物),A-23187 |
Apoptosis; Antibacterial; Antibiotic; Autophagy; Antifungal | Apoptosis; Autophagy; Microbiology/Virology |
Calcimycin (A-23187) 是抗生素和二价阳离子离子载体。它抑制革兰氏阳性细菌和一些真菌生长,也抑制 ATP 酶的活性并解耦哺乳动物细胞的氧化磷酸化。它通过增加细胞内钙浓度诱导 Ca2+依赖性细胞死亡。 | |||
TQ0251 |
(Z)-2-decenoic acid
(Z)-dec-2-enoic acid,(Z)-2-癸烯酸,cis-2-Decenoic acid,cis-dec-2-enoic acid |
Others | Others |
(Z)-2-decenoic acid (cis-dec-2-enoic acid) 是一种由铜绿假单胞菌产生的不饱和脂肪酸。它能够诱导一系列革兰氏阴性细菌(包括铜绿假单胞菌)和革兰氏阳性细菌形成的生物膜发生分散反应。它能够抑制生物膜发育。 | |||
T8247 |
(+)-Aromadendrene
|
Anti-infection | Microbiology/Virology |
(+)-Aromadendrene 是一种天然产物,对革兰氏阳性菌和革兰氏阴性菌具有显着的抗菌活性。 | |||
T1665 |
Daptomycin
达托霉素,LY146032 |
DNA/RNA Synthesis; Antibacterial; Antibiotic | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology |
Daptomycin (LY146032) 是脂肽类抗生素,在体外快速灭活革兰氏阳性细菌。 | |||
T8062 |
Cefazedone
Refosporen,头孢西酮 |
Others; Antibacterial; Antibiotic | Microbiology/Virology; Others |
Cefazedone (Refosporen) 是一种具有抗革兰氏阳性和革兰氏阴性菌活性的时间依赖性头孢菌素抗生素。 | |||
TN2279 |
Totarol
(+)-Totarol,桃柁酚 |
Antibacterial; Antifection | Microbiology/Virology |
Totarol ((+)-Totarol) 对几种致病性革兰氏阳性细菌、结核分枝杆菌具有抗菌作用。 | |||
T1134 |
Clofoctol
叔辛酚氯,氯福克酚 |
Antibacterial; Antibiotic | Microbiology/Virology |
Clofoctol 是一种抗生素,,可研究革兰氏阳性菌感染。它仅对革兰氏阳性菌起作用, 可渗透入人类肺组织。 | |||
T5037 |
Midecamycin
Antibiotic SF-837,Turimycin P3,Medecamycin A1,Rubimycin,麦迪霉素,Platenomycin B1,Espinomycin A |
Antibacterial; Antibiotic | Microbiology/Virology |
Midecamycin (Medecamycin A1) 是乙酰氧基取代的大环内酯类抗生素,对革兰氏阳性和阴性菌有效。 | |||
T1306 |
Norfloxacin
氟哌酸,MK-0366,诺氟沙星 |
DNA gyrase; Topoisomerase; Endogenous Metabolite; Antibacterial; Antibiotic | DNA Damage/DNA Repair; Metabolism; Microbiology/Virology |
Norfloxacin (MK-0366) 是广谱抗生素,能通过结合DNA 旋转酶抑制革兰氏阳性和阴性菌。 | |||
T1679 |
Thiostrepton
Thiactin,Bryamycin,Alaninamide,硫链丝菌素 |
DNA/RNA Synthesis; Antibacterial; Antibiotic | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology |
Thiostrepton (Alaninamide) 是一种选择性抑制FOXM1的抗生素。FOXM1会与 YAP/TEAD 复合物结合,形成YAP/TEAD/FOXM1 复合物。 | |||
T8302 |
Ceftiofur
|
Antibacterial; Antibiotic | Microbiology/Virology |
Ceftiofur 是一种半合成抗生素,对家畜的各种革兰氏阳性和革兰氏阴性菌、好氧菌和厌氧菌均有抗菌活性。 | |||
T0814L |
Ampicillin
Amcill,D-(-)-α-Aminobenzylpenicillin,Aminobenzylpenicillin,氨苄青霉素,Ampicillin acid |
Antibacterial; Antibiotic | Microbiology/Virology |
Ampicillin (Aminobenzylpenicillin) 属于 β-内酰胺类抗生素,是一种半合成的青霉素。Ampicillin 具有杀菌活性,对各种革兰氏阳性细菌和革兰氏阴性细菌均有抑制活性。 | |||
T5S0814 |
Berberine hydrogen sulphate
Berberine Bisulfate,硫酸氢黄连素,Umbellatine Sulfate |
Antibacterial | Microbiology/Virology |
Berberine hydrogen sulphate (Umbellatine Sulfate) 是一种从几种植物中提取的生物碱,对多种微生物具有抗菌活性,包括革兰氏阳性和革兰氏阴性细菌、真菌和原生动物。 | |||
T5274 |
D-(+)-Phenyllactic acid
D-3-苯乳酸,D-3-Phenyllactic acid |
Endogenous Metabolite; Antibacterial | Metabolism; Microbiology/Virology |
D-(+)-Phenyllactic acid (D-3-Phenyllactic acid) 是一种由白地霉分泌得到的抗菌剂,可抑制部分来自人类和食品的革兰氏阳性菌以及来自人类的革兰氏阴性菌。 | |||
T8504 |
Dianemycin
Nanchangmycin (free acid) |
Antibacterial; Antibiotic | Microbiology/Virology |
Dianemycin (Nanchangmycin (free acid)) 由Streptomyces nanchangensis 产生的一种聚醚抗生素,抑制革兰氏阳性菌。它也是一种针对 Zika 病毒的广谱抗病毒药物。 | |||
T5003 |
Rifamycin sodium
Rifamycin sodium salt,利福霉素钠 |
Antibacterial; Antibiotic | Microbiology/Virology |
Rifamycin sodium (Rifamycin sodium salt) salt 是从地中海曲霉或其突变体的发酵中分离出来的一种安沙霉素抗生素家族。它对革兰氏阳性菌和某些革兰氏阴性菌有抗生素活性。 | |||
TN1651 |
Furanodiene
|
Apoptosis; PARP; Reactive Oxygen Species; Caspase; CDK; P-gp | Apoptosis; Cell Cycle/Checkpoint; Chromatin/Epigenetic; DNA Damage/DNA Repair; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience; NF-κB; Proteases/Proteasome |
Furanodiene 是从姜黄中提取的一种萜类天然产物,可抑制外排转运蛋白Pgp 功能并降低 Pgp 蛋白水平。它通过抗血管生成和诱导ROS 产生,DNA 链断裂和细胞凋亡发挥抗癌作用。 | |||
T0906 |
Salinomycin
盐霉素,Procoxacin |
Wnt/beta-catenin; Antibacterial | Cytoskeletal Signaling; Microbiology/Virology; Stem Cells |
Salinomycin (Procoxacin)是一种多醚类钾离子载体抗生素,特异性抑制革兰氏阳性细菌生长。Salinomycin 作为Wnt/β-连环蛋白信号通路的有效抑制剂,阻断Wnt诱导的LRP6磷酸化。此外,Salinomycin (Procoxacin)对人类癌症干细胞显示出选择性活性。 | |||
T0958 |
Penicillin G sodium salt
青霉素钠,Penicillin G Sodium,Benzylpenicillin sodium salt,Benzylpenicillin Sodium |
GABA Receptor; Antibacterial; Antibiotic | Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience |
Penicillin G sodium(Benzylpenicillin sodium) salt 是一种 β-内酰胺类抗生素。 | |||
T12830 |
Sapienic acid sodium
|
Antibacterial | Microbiology/Virology |
Sapienic acid sodium,主要存在于皮肤和粘膜中的脂肪酸,对皮肤和口腔内的革兰氏阳性及阴性细菌展现出不同程度的抗菌效果。其对血链球菌、微生物链球菌与核纤梭菌的抗菌活性表现,MBC值分别为31.3 μg/mL、375.0 μg/mL与93.8 μg/mL。 | |||
T20643 |
Cefoxitin
Rephoxitin,Cefoxitinum |
Cell wall; Antibacterial; Antibiotic | Immunology/Inflammation; Microbiology/Virology |
Cefoxitin (Rephoxitin) 是一种广谱的、可口服的第二代头孢霉素类抗生素。Cefoxitin 干扰细菌细胞壁的合成。其活性谱包括革兰氏阴性和革兰氏阳性菌,通常用于腹腔感染、盆腔感染和某些类型的妇科感染等腹部,对厌氧菌具有高效性。 | |||
TN7231 |
Di-O-methylhonokiol
Honokiol dimethyl ether |
Antioxidant | oxidation-reduction |
Di-O-methylhonokiol (Honokiol dimethyl ether) 是Magnolia grandiflora L 的酚类成分,具有抗微生物活性,对革兰氏阳性和抗酸细菌和真菌具有显著的抗氧化活性。 | |||
T2989 |
4-Hydroxybenzoic acid
p-hydroxybenzoic acid,para-Hydroxybenzoic acid,PHBA,对羟基苯甲酸,4-hydroxybenzoate |
Endogenous Metabolite; Antibacterial | Metabolism; Microbiology/Virology |
4-Hydroxybenzoic acid (4-hydroxybenzoate) 是苯甲酸的酚衍生物,可抑制革兰氏阳性和革兰氏阴性菌,IC50值为160 μg/mL。 | |||
T4S0867 |
Pogostone
DHELWANGIN,广藿香酮 |
Apoptosis; Antibacterial; Autophagy | Apoptosis; Autophagy; Microbiology/Virology |
Pogostone (DHELWANGIN) 是从薄荷中分离出,对革兰氏阴性菌、革兰氏阳性菌、大肠埃希菌等具有强效抗菌、抗真菌活性。它诱导细胞凋亡和自噬。 | |||
T8347 |
Rifamycin S
|
Reactive Oxygen Species; ROS; Antibacterial; Antibiotic | Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB |
Rifamycin S 是一种 DNA 依赖性 RNA 聚合酶抑制剂,是一种醌和一种针对革兰氏阳性细菌的抗生素试剂。它是涉及两个电子的可逆氧化还原系统的氧化形式。它能产生活性氧并抑制微粒体脂质过氧化,可研究肺结核和麻风病。 | |||
T1219 |
Sisomicin Sulfate
硫酸西索米星,Pathomycin,Extramycin,硫酸西索紫苏 |
Antibacterial; Antibiotic | Microbiology/Virology |
Sisomicin Sulfate (Pathomycin) 是由Micromonospora inyoensis 产生的一种广谱氨基糖苷类抗生素,对革兰氏阳性细菌有很大活性。 | |||
T3092 |
Nigericin sodium salt
尼日利亚菌素,尼日利亚菌素钠盐 |
Potassium Channel; NOD-like Receptor (NLR); Antibacterial; Antibiotic; NOD | Immunology/Inflammation; Membrane transporter/Ion channel; Microbiology/Virology; NF-κB |
Nigericin sodium salt 属于抗生素,是一种 NLRP3 激活剂,也是一种阳离子离子载体。Nigericin sodium 可以触发 NALP3 炎性体的激活,可抑制高尔基体功能并抑制革兰氏阳性菌的生长。 | |||
T0819 |
Spiramycin
Espiramicin,螺旋霉素,Sequamycin,Rovamycin,Provamycin,Formacidine |
Antibacterial; Antibiotic; Parasite | Microbiology/Virology |
Spiramycin (Rovamycin) 是一种由安博链霉菌产生的大环内酯类抗生素,具有抗细菌和弓形虫活性,并具有抗寄生虫作用。它由 16 个内酯环组成,其上附着 mycaminose,forosamine 和 mycarose 三种糖。 | |||
T4S1943 |
Kirenol
奇壬醇,奇任醇,Kirel |
Wnt/beta-catenin | Cytoskeletal Signaling; Stem Cells |
Kirenol (Kirel) 是分离自 Siegesbeckia orientalis 中的,具有抗氧化、抗炎、抗过敏、抗关节炎活性,可用于缓解疼痛的研究。 | |||
T26805 |
Bicyclomycin
Bicozamycin |
||
Bicyclomycin is a broad spectrum antibiotic active against Gram-negative bacteria and the Gram-positive bacterium, Micrococcus luteusn. | |||
TN4518 |
Meridinol
|
Antifection | Microbiology/Virology |
Meridinol has wide antimicrobial activity, includes against gram-positive and gram-negative bacteria and fungi. | |||
T11551 |
Helvolic acid
Fumigacin |
Others | Others |
Helvolic acid, an antibiotic derived from Xylaria sp., exhibits effectiveness against Gram-positive bacteria. | |||
TN6002 |
Crenatine
1-Ethyl-4-methoxy-β-carboline |
||
Crenatine possesses antibacterial activity, it is more effective against Gram-positive than Gram-negative bacteria. | |||
T27024 |
Citromycetin
Frequentic Acid,NSC-53584,NSC 53584,NSC53584 |
||
Citromycetin is a fungal metabolite originally isolated from Australian P. frequentans. It has antibiotic activity against the Gram-negative bacteria V. cholerae and S. flexneri and the Gram-positive bacteria S. aureus. | |||
T38176 |
Muramic acid
|
||
Muramic acid is a prevalent constituent found in the cell walls of Gram-positive bacteria, serving as a distinguishing marker for such bacteria[1]. | |||
TN1301 |
6,8-Diprenylgenistein
6,8-二异戊烯基金雀异黄素,鲁冰花 |
Antifection | Microbiology/Virology |
6,8-Diprenylgenistein has antimicrobial activity, it has anti-bacteria activity against Gram-negative and Gram-positive bacteria. | |||
T4131 | Arjunic acid | COX; Antifection | Immunology/Inflammation; Microbiology/Virology; Neuroscience |
Arjunic acid is a strong antioxidant and a free radical scavenger. Arjunic acid shows activity against Gram-positive and Gram-negative bacteria with MIC values ranging between 1.9 and 15.6 microg/mL. | |||
TN6163 |
3-O-cis-p-Coumaroylmaslinic acid
|
||
3-beta-O-(trans-p-Coumaroyl)maslinic acid shows antimicrobial activity on Gram-positive bacteria and yeasts. | |||
TN2502 | 1,5,6-Trihydroxyxanthone | Others | Others |
1,5,6-Trihydroxyxanthone exhibits antibacterial activity against Gram-positive bacteria. | |||
TN4264 |
Isoapetalic acid
胡桐,海棠木 |
HIV Protease; Antifection | Microbiology/Virology; Proteases/Proteasome |
Isoapetalic acid and apetalic acid exhibit cytotoxic activities towards both cancer cell lines(human breast cancer (MCF-7) and human lung carcinoma (A-549) cell lines) and both Gram-positive bacteria(two Gram-positive bacteria, S. aureus and B. subtilis a | |||
T16673 |
Pseudouridimycin
PUM |
Others | Others |
Pseudouridimycin is a C-nucleoside analogue. Pseudouridimycin is an antibiotic and is a selective bacterial RNA polymerase (RNAP) inhibitor. It is effective against both Gram-negative and Gram-positive bacteria. | |||
TN6148 |
3-O-trans-p-Coumaroylmaslinic acid
|
||
3-beta-O-(trans-p-Coumaroyl)maslinic acid is a DNA polymerase B" inhibitor. It shows antimicrobial activity on Gram-positive bacteria and yeasts. | |||
TN5930 |
Ocotillone
|
||
Ocotillone has potent antibacterial activity against Gram-negative bacteria, P. aeruginosa and S. typhimurium, that are without hemolytic activity, whereas it has weak antimicrobial activity against Gram-positive bacteria and fungi. Ocotillone shows only | |||
T32924 |
Lucidin ethyl ether
|
||
Ibericin 是一种从Prismatomeris filamentosa 根中分离得到的蒽醌代谢产物,对革兰氏阳性菌和革兰氏阴性菌具有一定的抗菌活性。 | |||
T71909 |
Kumbicin C
|
||
Kumbicin C inhibits the growth of NS-1 mouse myeloma cells (IC50 = 0.74 μg/ml) and the growth of the Gram-positive bacteria B. subtilis (MIC = 1.6 μg/ml). | |||
T10455 |
Bafilomycin B1
巴佛洛霉素 B1 |
Others | Others |
Bafilomycin B1, a macrolide antibiotic isolated from Streptomyces sp, acts as an inhibitor of K+-dependent ATPase of E. coli. It also inhibits Gram-positive bacteria and fungi. | |||
T27977 |
Manzamine A
Keramamine A |
||
Manzamine A is a GSK-3 inhibitor and vacuolar ATPase uncoupler found in marine sponges. It inhibits autophagy and tumor growth in cancer models, suppresses foam cell formation in macrophages, prevents growth of gram negative and gram positive bacteria, an | |||
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